SCHEMBL4044026

SCHEMBL4044026

CC(C)CC(NC(=O)Oc1ccoc1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1ccccn1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSK P43235 18/20 0.49
CTSL P07711 8/20 0.45
CTSS P25774 7/20 0.45
KDM4E B2RXH2 2/20 0.37
ALDH1A1 P00352 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CTSB P07858 2/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050717 0.92 CTSK (0.44) CTSKCTSLCTSS
SCHEMBL4049845 0.92 CTSK (0.40) CTSKCTSLCTSS
SCHEMBL4041369 0.89 CTSS (0.42) CTSKCTSLCTSS
SCHEMBL4045333 0.89 CTSK (0.53) CTSKCTSLCTSSKDM4EALDH1A1
SCHEMBL4047693 0.88 CTSK (0.40) CTSKCTSLCTSSKDM4EALDH1A1
SCHEMBL4046943 0.87 CTSK (0.50) CTSKCTSLCTSSKDM4EALDH1A1
SCHEMBL4045548 0.87 CTSK (0.51) CTSKCTSLCTSSKDM4EALDH1A1
SCHEMBL4042251 0.87 CTSK (0.50) CTSKCTSLCTSSKDM4EALDH1A1
SCHEMBL4043401 0.85 CTSK (0.47) CTSKCTSLCTSSKDM4EALDH1A1
SCHEMBL4043679 0.85 CTSK (0.46) CTSKCTSLCTSSCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed