SCHEMBL4044582

SCHEMBL4044582

CCCC(NC(=O)Oc1ccc2ccccc2n1)C(=O)N1CCC2C1C(=O)CN2C(=O)c1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.40
PREP P48147 4/20 0.38
FAP Q12884 4/20 0.38
CTSL P07711 3/20 0.35
CTSS P25774 3/20 0.35
CTSB P07858 1/20 0.35
MC4R P32245 1/20 0.34
MC3R P41968 1/20 0.34
MC1R Q01726 1/20 0.34
PDE5A O76074 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE7A Q13946 1/20 0.33
PDE3A Q14432 1/20 0.33
TGM2 P21980 1/20 0.32
HTR1A P08908 2/20 0.31
DRD2 P14416 2/20 0.31
HTR7 P34969 2/20 0.31
HTR6 P50406 2/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041452 0.92 CTSK (0.49) CTSKCTSLCTSSCTSBKDM4E
SCHEMBL4042489 0.91 CTSK (0.40) CTSKPREPFAPCTSLCTSS
SCHEMBL4043597 0.88 CTSK (0.41) CTSKPREPFAPCTSLCTSS
SCHEMBL4052232 0.88 CTSK (0.38) CTSKPREPFAPCTSLCTSS
SCHEMBL6237514 0.88 CTSK (0.46) CTSKPREPFAPCTSLCTSS
SCHEMBL4049188 0.86 CTSK (0.40) CTSKPREPFAPCTSLCTSS
SCHEMBL4044872 0.86 CTSK (0.44) CTSKPREPFAPCTSLCTSS
SCHEMBL4043756 0.85 CTSK (0.40) CTSKPREPFAPCTSLCTSS
SCHEMBL4045843 0.85 CTSK (0.43) CTSKPREPFAPCTSLCTSS
SCHEMBL4045942 0.84 CTSK (0.41) CTSKPREPFAPCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed