SCHEMBL4044689

SCHEMBL4044689

CCCC(NC(=O)Oc1ccco1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
CTSK P43235 16/20 0.35
CTSL P07711 13/20 0.35
CTSS P25774 12/20 0.35
ELANE P08246 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050718 0.92 CTSK (0.41) CTSKCTSLCTSSALDH1A1
SCHEMBL4044283 0.89 CTSK (0.45) CTSKCTSLCTSS
SCHEMBL4047765 0.88 PREP (0.35) PREPFAPCTSKCTSLCTSS
SCHEMBL6235917 0.88 CTSK (0.46) PREPFAPCTSKCTSLCTSS
SCHEMBL4048824 0.88 CTSK (0.37) PREPFAPCTSKCTSLCTSS
SCHEMBL4042961 0.88 CTSK (0.36) PREPFAPCTSKCTSLCTSS
SCHEMBL4043139 0.87 ELANE (0.37) PREPFAPCTSKELANEALDH1A1
SCHEMBL4051063 0.87 SMYD3 (0.36) PREPFAPCTSKCTSLCTSS
SCHEMBL4038257 0.87 PREP (0.34) PREPFAPCTSKELANEALDH1A1
SCHEMBL4045026 0.86 CTSK (0.36) PREPFAPCTSKCTSLCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1463728-B1 FUSED CYCLIC MODULATORS OF NUCLEAR HORMONE RECEPTOR FUNCTION BRISTOL MYERS SQUIBB CO (US) 2009-01-14 EP disclosed