SCHEMBL4047765

SCHEMBL4047765

CCCC(NC(=O)Oc1ccoc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
ELANE P08246 1/20 0.33
CTSK P43235 5/20 0.33
CTSL P07711 3/20 0.31
CTSS P25774 3/20 0.31
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049692 0.93 CTSK (0.37) ELANECTSKCTSLCTSSKMT2A
SCHEMBL4045340 0.92 CTSK (0.40) ELANECTSKCTSLCTSSALDH1A1
SCHEMBL4043139 0.90 ELANE (0.37) PREPFAPELANECTSKALDH1A1
SCHEMBL4046656 0.90 CTSK (0.40) CTSKCTSLCTSS
SCHEMBL4044689 0.88 PREP (0.35) PREPFAPELANECTSKCTSL
SCHEMBL4045026 0.88 CTSK (0.36) PREPFAPELANECTSKCTSL
SCHEMBL4047831 0.88 PREP (0.35) PREPFAPELANECTSKALDH1A1
SCHEMBL4041785 0.88 PREP (0.35) PREPFAPCTSKCTSLCTSS
SCHEMBL4047173 0.87 SMYD3 (0.35) PREPFAPALDH1A1
SCHEMBL4048179 0.87 TSHR (0.36) PREPFAPELANEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed