SCHEMBL4044904

SCHEMBL4044904

NC(=O)C(CNC[C@@H](O)[CH]Cc1ccccc1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 3/20 0.51
BCAT2 O15382 1/20 0.40
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ABCB1 P08183 2/20 0.37
CNR2 P34972 1/20 0.37
BCHE P06276 1/20 0.36
POLB P06746 1/20 0.35
CYP2C19 P33261 1/20 0.35
CNR1 P21554 1/20 0.35
UBE2N P61088 1/20 0.35
CRHBP P24387 1/20 0.35
CRHR2 Q13324 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4047002 0.80 EPHX1 (0.42) EPHX1BCAT2ABCB1CNR2
SCHEMBL7054852 0.78 ALDH1A1 (0.47) KDM4EL3MBTL1
SCHEMBL3939381 0.77 BCHE (0.47) BCHE
SCHEMBL27598444 0.75 HPGD (0.42) KDM4EL3MBTL1
SCHEMBL5219600 0.75 ANPEP (0.46) BCHE
SCHEMBL4039140 0.74 ABCB1 (0.47) KDM4EABCB1BCHECYP2C19CNR1
SCHEMBL7616171 0.73 EPHX1 (0.54) EPHX1BCAT2KDM4EL3MBTL1CNR2
SCHEMBL4045031 0.73 KDM1A (0.46) BCHE
SCHEMBL4043818 0.73 BCHE (0.41) BCHE
SCHEMBL4041830 0.72 METAP2 (0.41) KDM4ECNR2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678157-A4 HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THEREOF REDDY US THERAPEUTICS INC (US) 2009-03-18 EP disclosed
EP-1678157-A2 HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THEREOF Reddy US Therapeutics, Inc. (US) 2006-07-12 EP disclosed
WO-2005042712-A2 HETEROCYCLIC COMPOUNDS AND METHODS OF MAKING AND USING THEREOF REDDY US THERAPEUTICS, INC. (US) 2005-05-12 WO disclosed