SCHEMBL4045215

SCHEMBL4045215

O=C(O)c1c(Cl)c(-c2cccnc2)n2c1CN(S(=O)(=O)c1ccc(C(F)(F)F)cc1)CC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.43
GBA1 P04062 2/20 0.41
L3MBTL1 Q9Y468 3/20 0.40
HSD11B1 P28845 2/20 0.40
LMNA P02545 1/20 0.40
NAMPT P43490 2/20 0.39
CYP3A4 P08684 3/20 0.39
CYP2D6 P10635 1/20 0.39
GCK P35557 1/20 0.39
CCR6 P51684 1/20 0.38
ABL1 P00519 1/20 0.38
BCR P11274 1/20 0.38
P2RX7 Q99572 1/20 0.38
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC7 Q8WUI4 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC10 Q969S8 1/20 0.37
HDAC11 Q96DB2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036841 0.92 CYP11B1 (0.42) CYP11B1GBA1L3MBTL1HSD11B1LMNA
SCHEMBL4036720 0.83 GBA1 (0.43) GBA1L3MBTL1LMNACYP2D6GCK
SCHEMBL14394007 0.81 CYP11B1 (0.41) CYP11B1GBA1L3MBTL1HSD11B1LMNA
SCHEMBL6658946 0.76 P2RX7 (0.41) ABL1BCRP2RX7
SCHEMBL4047940 0.76 LSS (0.37) GBA1CYP3A4CYP2D6USP2
SCHEMBL6632666 0.75 LMNA (0.47) GBA1HSD11B1LMNACYP3A4CYP2D6
SCHEMBL4037080 0.73 HTT (0.48) GBA1LMNAALDH1A1USP2GAA
SCHEMBL14393987 0.72 TRPV1 (0.52)
SCHEMBL4041961 0.72 PKM (0.47) GBA1ALDH1A1USP2GAAHPGD
SCHEMBL4044206 0.72 KMT2A (0.42) ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1436291-B1 INDOLIZINES AS KINASE PROTEIN INHIBITORS AVENTIS PHARMA SA (FR) 2009-01-14 EP disclosed