SCHEMBL4045745

SCHEMBL4045745

COc1cc(N)cc(OCCN(C)C)c1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.49
FYN P06241 2/20 0.48
AOC3 Q16853 2/20 0.46
LMNA P02545 1/20 0.45
DRD2 P14416 1/20 0.45
ACHE P22303 1/20 0.45
SLC6A2 P23975 1/20 0.45
CYP2C19 P33261 1/20 0.45
DRD3 P35462 1/20 0.45
KCNH2 Q12809 1/20 0.45
NOS3 P29474 2/20 0.45
NOS1 P29475 2/20 0.45
MAPK1 P28482 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP19A1 P11511 2/20 0.42
KDM4E B2RXH2 2/20 0.40
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
HTR2A P28223 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4036416 0.92 FYN (0.53) HTR7FYNAOC3LMNADRD2
SCHEMBL4041993 0.84 CYP2D6 (0.46) AOC3DRD2DRD3SMN1; SMN2ALDH1A1
SCHEMBL8188932 0.83 HTR7 (0.49) HTR7FYNAOC3LMNADRD2
SCHEMBL1220219 0.80 HTR7 (0.53) HTR7DRD2DRD3NOS3NOS1
SCHEMBL5275674 0.80 GAA (0.60) HTR7ACHENOS3NOS1MAPK1
SCHEMBL29875923 0.80 GAA (0.60) HTR7ACHENOS3NOS1MAPK1
SCHEMBL191996 0.78 ACHE (0.59) ACHEMAPK1CYP19A1KDM4EGAA
SCHEMBL21048199 0.76 ROCK2 (0.43) HTR7DRD2NOS3NOS1ALDH1A1
SCHEMBL19732163 0.76 HTR7 (0.51) HTR7FYNNOS3NOS1ALDH1A1
SCHEMBL7955166 0.75 FYN (0.47) HTR7FYNAOC3LMNADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562589-B1 DIAMINOTRIAZOLES USEFUL AS INHIBITORS OF PROTEIN KINASES VERTEX PHARMA (US) 2009-01-07 EP disclosed