SCHEMBL4045797

SCHEMBL4045797

Cc1cc(Br)ccc1-c1ncc(Br)o1.Cc1cc(Br)ccc1C1=NCCO1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
NPC1 O15118 1/20 0.32
TSHR P16473 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4500247 0.85 SMN1; SMN2 (0.38) CRHR1SMN1; SMN2NPC1TSHRRAB9A
SCHEMBL3953788 0.84 NPC1 (0.37) CRHR1SMN1; SMN2NPC1TSHRRAB9A
SCHEMBL4044503 0.77 SMN1; SMN2 (0.35) CRHR1SMN1; SMN2
SCHEMBL6515580 0.71 LMNA (0.43) SMN1; SMN2NPC1RAB9A
SCHEMBL9668468 0.68 ESR2 (0.47) SMN1; SMN2
SCHEMBL25194674 0.68 SMN1; SMN2 (0.36) SMN1; SMN2NPC1TSHRRAB9A
SCHEMBL7957225 0.66 GABRA1 (0.35) SMN1; SMN2NPC1
SCHEMBL25211116 0.66 SMN1; SMN2 (0.38) SMN1; SMN2NPC1RAB9A
SCHEMBL1842317 0.64 SMN1; SMN2 (0.48) SMN1; SMN2NPC1TSHRRAB9A
SCHEMBL25193298 0.63 SMN1; SMN2 (0.40) SMN1; SMN2NPC1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697333-A4 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-1697333-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS Merck & Co., Inc. (US) 2006-09-06 EP disclosed
WO-2005058848-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO., INC. (US) 2005-06-30 WO disclosed