SCHEMBL4044503

SCHEMBL4044503

Cc1cc(Br)ccc1C1=NCCO1.O=C(Cl)C(=O)Cl

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.35
HPGD P15428 1/20 0.34
HTT P42858 1/20 0.34
MMP13 P45452 1/20 0.34
POLB P06746 1/20 0.33
P2RX4 Q99571 1/20 0.32
CRHR1 P34998 1/20 0.31
FFAR1 O14842 1/20 0.31
MAPT P10636 1/20 0.31
TUBB4A P04350 1/20 0.31
TUBB P07437 1/20 0.31
TUBA3C P0DPH7 1/20 0.31
TUBA1B P68363 1/20 0.31
TUBA4A P68366 1/20 0.31
TUBB4B P68371 1/20 0.31
TUBB3 Q13509 1/20 0.31
TUBB2A Q13885 1/20 0.31
TUBB8 Q3ZCM7 1/20 0.31
TUBA3E Q6PEY2 1/20 0.31
TUBA1A Q71U36 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4500247 0.90 SMN1; SMN2 (0.38) SMN1; SMN2HPGDHTTMMP13POLB
SCHEMBL4045797 0.77 CRHR1 (0.33) SMN1; SMN2CRHR1
SCHEMBL9668468 0.75 ESR2 (0.47) SMN1; SMN2MAPTALDH1A1
SCHEMBL6515580 0.75 LMNA (0.43) SMN1; SMN2HPGDMAPTALDH1A1
SCHEMBL25194674 0.71 SMN1; SMN2 (0.36) SMN1; SMN2HPGDHTTMMP13MAPT
SCHEMBL7957225 0.69 GABRA1 (0.35) SMN1; SMN2HPGDHTTMAPT
SCHEMBL25211116 0.69 SMN1; SMN2 (0.38) SMN1; SMN2MMP13MAPTALDH1A1
SCHEMBL1842317 0.68 SMN1; SMN2 (0.48) SMN1; SMN2HPGDALDH1A1
SCHEMBL7832365 0.67 ADH5 (0.45) ALDH1A1
SCHEMBL25193298 0.66 SMN1; SMN2 (0.40) SMN1; SMN2HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697333-A4 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO INC (US) 2009-07-08 EP disclosed
EP-1697333-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS Merck & Co., Inc. (US) 2006-09-06 EP disclosed
WO-2005058848-A1 (3,4-DISUBSTITUTED)PROPANOIC CARBOXYLATES AS S1P (EDG) RECEPTOR AGONISTS MERCK & CO., INC. (US) 2005-06-30 WO disclosed