SCHEMBL4045987

SCHEMBL4045987

CCOC(=O)Oc1cc2c(s1)-c1ccc(OCCN(C)C)cc1Oc1ccccc1-2

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
PDK2 Q15119 3/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HPGD P15428 1/20 0.37
MAOB P27338 2/20 0.36
CACNA1H O95180 1/20 0.36
CACNA1B Q00975 1/20 0.36
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
CYP3A4 P08684 1/20 0.36
BCHE P06276 1/20 0.35
MAOA P21397 1/20 0.35
ACHE P22303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041725 0.96 CACNA1B (0.41) HDAC3HDAC1HDAC2PDK2KDM4E
SCHEMBL4050340 0.89 CACNA1B (0.42) HDAC3HDAC1HDAC2PDK2KDM4E
SCHEMBL4043160 0.85 PPARG (0.43) ALDH1A1MEN1KMT2AHPGDMAOB
SCHEMBL4048452 0.85 MEN1 (0.43) HDAC3HDAC1HDAC2PDK2KDM4E
SCHEMBL4051251 0.84 ACHE (0.44) MAOBACHE
SCHEMBL4046658 0.84 CACNA1B (0.44) HDAC3HDAC1HDAC2PDK2KDM4E
SCHEMBL4044883 0.81 CACNA1B (0.43) HDAC3HDAC1HDAC2PDK2KDM4E
SCHEMBL6204224 0.81 TYMS (0.37) KDM4EALDH1A1MEN1KMT2AHPGD
SCHEMBL4047340 0.79 PPARG (0.44) ALDH1A1MEN1KMT2AMAOBMAOA
SCHEMBL5435148 0.77 KDM4E (0.44) HDAC3HDAC1HDAC2PDK2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1603921-B1 THIADIBENZOAZULENE DERIVATIVES FOR THE TREATMENT OF INFLAMMATORY DISEASES GLAXOSMITHKLINE ZAGREB (HR) 2009-06-17 EP claimed