SCHEMBL6204224

SCHEMBL6204224

CCOC(=O)Oc1cc2c(s1)-c1cc3ccccc3cc1Oc1ccccc1-2

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TYMS P04818 1/20 0.37
ALDH1A1 P00352 8/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
ALOX5 P09917 2/20 0.34
MAPT P10636 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
RXFP1 Q9HBX9 2/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 3/20 0.34
TDP1 Q9NUW8 1/20 0.34
GLA P06280 2/20 0.33
CA2 P00918 1/20 0.33
MEN1 O00255 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
RAB9A P51151 1/20 0.32
CTDSP1 Q9GZU7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6204660 0.91 MAOB (0.36) TYMSALDH1A1L3MBTL1MAPTKDM4E
SCHEMBL6204171 0.85 ALDH1A1 (0.38) TYMSALDH1A1L3MBTL1ALOX5MAPT
SCHEMBL6204597 0.83 ALDH1A1 (0.39) TYMSALDH1A1L3MBTL1MAPTKDM4E
SCHEMBL4047340 0.83 PPARG (0.44) ALDH1A1L3MBTL1KMT2ACA2MEN1
SCHEMBL4043160 0.82 PPARG (0.43) ALDH1A1L3MBTL1HPGDKMT2AMEN1
SCHEMBL5422453 0.82 ALDH1A1 (0.50) ALDH1A1L3MBTL1MAPTKDM4EHPGD
SCHEMBL4045987 0.81 HDAC3 (0.41) ALDH1A1KDM4EHPGDKMT2AMEN1
SCHEMBL4050340 0.81 CACNA1B (0.42) TYMSALDH1A1KDM4ESMN1; SMN2
SCHEMBL4041725 0.80 CACNA1B (0.41) ALDH1A1KDM4EKMT2AMEN1SMN1; SMN2
SCHEMBL6202961 0.79 LMNA (0.39) ALDH1A1L3MBTL1ALOX5MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1492795-B1 1- OR 3-THIA-BENZONAPHTHOAZULENES AS INHIBITORS OF TUMOUR NECROSIS FACTOR PRODUCTION AND INTERMEDIATES FOR THE PREPARATION THEREOF PLIVA ISTRAZIVACKI INST D O O (HR) 2005-11-16 EP claimed