SCHEMBL4045995

SCHEMBL4045995

CS(=O)(=O)C(N)c1cccc(-c2ccc(OC(F)(F)F)c(C(=O)O)c2)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
F2 P00734 3/20 0.40
F3 P13726 3/20 0.40
CFD P00746 1/20 0.39
DHODH Q02127 2/20 0.38
PTPN11 Q06124 2/20 0.38
RXRA P19793 1/20 0.37
RXRB P28702 1/20 0.37
RXRG P48443 1/20 0.37
CTSA P10619 3/20 0.37
F9 P00740 1/20 0.36
AKR1C2 P52895 1/20 0.35
AKR1C1 Q04828 1/20 0.35
KCNK3 O14649 2/20 0.35
KCNK9 Q9NPC2 2/20 0.35
ACLY P53396 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4026660 0.78 ACMSD (0.55) CFDDHODHPTPN11AKR1C2AKR1C1
SCHEMBL4040652 0.77 KIF11 (0.55)
SCHEMBL3947686 0.77 MCL1 (0.58) CFDDHODHPTPN11AKR1C2AKR1C1
SCHEMBL3936487 0.76 DCLRE1B (0.51) CFDDHODHPTPN11AKR1C2AKR1C1
SCHEMBL3944255 0.76 ACMSD (0.45) CFDDHODHPTPN11AKR1C2AKR1C1
SCHEMBL4042656 0.75 PTPN11 (0.51) CFDPTPN11AKR1C2KCNK3KCNK9
SCHEMBL3946016 0.75 KDM4E (0.53) ROCK2ROCK1CFDDHODH
SCHEMBL3944259 0.75 SLC6A2 (0.44) CFDDHODHPTPN11
SCHEMBL4046170 0.74 DCLRE1B (0.50) CFDDHODHPTPN11RXRARXRB
SCHEMBL3937100 0.74 KDM4E (0.47) CFDRXRARXRBACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2020404-A1 Cyanomethyl substituted N-Acyl Tryptamines Bayer Schering Pharma Aktiengesellschaft (DE) 2009-02-04 EP disclosed