SCHEMBL4046170

SCHEMBL4046170

O=C(O)c1cc(-c2cccc(Cl)c2)ccc1OC(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DCLRE1B Q9H816 1/20 0.50
AKR1C2 P52895 1/20 0.47
AKR1C1 Q04828 1/20 0.47
DHODH Q02127 2/20 0.44
CFD P00746 1/20 0.44
KMO O15229 2/20 0.43
ACLY P53396 2/20 0.42
SLC6A9 P48067 1/20 0.42
ANO1 Q5XXA6 1/20 0.42
PTPN11 Q06124 1/20 0.41
HCAR2 Q8TDS4 1/20 0.41
ACMSD Q8TDX5 1/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
PTPN22 Q9Y2R2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1972984 0.87 AKR1C2 (0.53) AKR1C2AKR1C1DHODHCFDKMO
SCHEMBL4026660 0.87 ACMSD (0.55) DCLRE1BAKR1C2AKR1C1DHODHCFD
SCHEMBL3936487 0.84 DCLRE1B (0.51) DCLRE1BAKR1C2AKR1C1DHODHCFD
SCHEMBL3944255 0.84 ACMSD (0.45) AKR1C2AKR1C1DHODHCFDPTPN11
SCHEMBL2115556 0.84 TSHR (0.53) AKR1C2AKR1C1DHODHKMOANO1
SCHEMBL29646503 0.84 TSHR (0.53) AKR1C2AKR1C1DHODHKMOANO1
SCHEMBL3937100 0.83 KDM4E (0.47) CFDKMOACLYRXRARXRB
SCHEMBL3947686 0.83 MCL1 (0.58) AKR1C2AKR1C1DHODHCFDKMO
SCHEMBL4038391 0.81 ACMSD (0.60) DHODHCFDPTPN11ACMSD
SCHEMBL4042656 0.81 PTPN11 (0.51) AKR1C2CFDACLYPTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20090069321-A1 CYANOMETHYL SUBSTITUTED N-ACYL TRYPTAMINES BAYER SCHERING PHARMA AG (DE) 2009-03-12 US claimed
EP-2020404-A1 Cyanomethyl substituted N-Acyl Tryptamines Bayer Schering Pharma Aktiengesellschaft (DE) 2009-02-04 EP claimed
US-20090069321-A1 CYANOMETHYL SUBSTITUTED N-ACYL TRYPTAMINES BAYER SCHERING PHARMA AG (DE) 2009-03-12 US disclosed
EP-2020404-A1 Cyanomethyl substituted N-Acyl Tryptamines Bayer Schering Pharma Aktiengesellschaft (DE) 2009-02-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090069321-A1 CYANOMETHYL SUBSTITUTED N-ACYL TRYPTAMINES FSHR, GNRHR, HNMT DCLRE1B 4209/4885AKR1C2 1308/4885AKR1C1 1332/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.