SCHEMBL4046660

SCHEMBL4046660

CC(C)CC(NC(=O)Oc1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.40
RECQL P46063 1/20 0.40
ELOVL6 Q9H5J4 1/20 0.39
CTSK P43235 2/20 0.38
HSD17B10 Q99714 1/20 0.36
KCNQ1 P51787 2/20 0.35
HCRTR2 O43614 1/20 0.35
POLB P06746 1/20 0.34
PIK3CG P48736 1/20 0.34
TSHR P16473 3/20 0.34
LMNA P02545 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
GPR119 Q8TDV5 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
SMYD3 Q9H7B4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050093 0.93 HTT (0.41) HTTRECQLELOVL6HSD17B10KCNQ1
SCHEMBL4050939 0.90 CTSK (0.37) HTTRECQLCTSKPOLBTSHR
SCHEMBL4039972 0.90 CTSK (0.40) HTTRECQLCTSKPOLBTSHR
SCHEMBL4040677 0.89 CTSK (0.41) ELOVL6CTSKHSD17B10KCNQ1HCRTR2
SCHEMBL4047459 0.88 CTSK (0.38) CTSKKCNQ1TSHRLMNAALDH1A1
SCHEMBL4051777 0.87 CTSK (0.44) ELOVL6CTSKHSD17B10KCNQ1HCRTR2
SCHEMBL4045230 0.87 CTSK (0.43) ELOVL6CTSK
SCHEMBL4045961 0.86 CTSK (0.39) ELOVL6CTSKHSD17B10KCNQ1HCRTR2
SCHEMBL4049970 0.86 CTSK (0.40) ELOVL6CTSKHSD17B10KCNQ1HCRTR2
SCHEMBL4050084 0.85 CTSK (0.41) CTSKPOLBTSHRLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed