SCHEMBL4050084

SCHEMBL4050084

CC(C)CC(NC(=O)Oc1ccc2c(c1)OCO2)C(=O)N1CCC2C1C(=O)CN2C(=O)Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 5/20 0.41
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KMT2A Q03164 1/20 0.36
ESR2 Q92731 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
PAX8 Q06710 1/20 0.35
BMP1 P13497 1/20 0.35
EDNRA P25101 1/20 0.35
CTSL P07711 2/20 0.34
CTSB P07858 2/20 0.34
CHRNA7 P36544 2/20 0.34
CTSS P25774 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNA4 P43681 1/20 0.34
TSHR P16473 2/20 0.34
LMNA P02545 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046542 0.93 POLB (0.36) CTSKALDH1A1MEN1USP2POLB
SCHEMBL4045179 0.89 CTSK (0.44) CTSKPAX8CTSLCTSBCHRNA7
SCHEMBL4050939 0.87 CTSK (0.37) CTSKALDH1A1MEN1USP2POLB
SCHEMBL4045083 0.87 CTSK (0.47) CTSKCTSLCTSBCHRNA7CTSS
SCHEMBL4048629 0.86 CTSK (0.42) CTSKALDH1A1PAX8CTSLCTSB
SCHEMBL4050440 0.86 CTSK (0.43) CTSKALDH1A1PAX8CTSLCTSB
SCHEMBL4046660 0.85 HTT (0.40) CTSKALDH1A1POLBTSHRLMNA
SCHEMBL4049343 0.85 CTSK (0.43) CTSKALDH1A1PAX8CTSLCTSB
SCHEMBL4044450 0.84 CTSK (0.43) CTSKALDH1A1PAX8CTSLCTSB
SCHEMBL4039972 0.83 CTSK (0.40) CTSKALDH1A1MEN1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed