SCHEMBL4046829

SCHEMBL4046829

N#Cc1cccc2c1C=COO2

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.34
TSHR P16473 1/20 0.32
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481312 0.71 ALDH1A1 (0.33) KDM4EALDH1A1CA1CA2
SCHEMBL27612514 0.69 CYP2B6 (0.40) TRPA1TSHRKDM4EALDH1A1CA1
SCHEMBL15320699 0.67 TRPA1 (0.35) TRPA1
SCHEMBL4237083 0.67 DYRK1A (0.37) TRPA1TSHR
SCHEMBL286500 0.66 TRPA1 (0.33) TRPA1TSHRKDM4EALDH1A1CA1
SCHEMBL2965295 0.65 KDM4E (0.36) TRPA1KDM4EALDH1A1
SCHEMBL15320700 0.63 TRPA1 (0.38) TRPA1
SCHEMBL9618582 0.63
SCHEMBL4046834 0.63 TRPA1 (0.44) TRPA1TSHRCA1CA2
SCHEMBL7300186 0.62 ITGB2 (0.35) TRPA1TSHRKDM4EALDH1A1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2010532-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS Glaxo Group Limited (GB) 2009-01-07 EP claimed
WO-2007122258-A1 TRYCLIC NITROGEN CONTAINING COMPOUNDS AND THEIR USE AS ANTIBACTERIALS GLAXO GROUP LIMITED (GB) 2007-11-01 WO claimed