SCHEMBL4046923

SCHEMBL4046923

CCCCCc1nc2nccnc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PI4KA P42356 1/20 0.51
PI4K2B Q8TCG2 1/20 0.51
PI4K2A Q9BTU6 1/20 0.51
PI4KB Q9UBF8 1/20 0.51
GPR84 Q9NQS5 5/20 0.44
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
HCAR2 Q8TDS4 1/20 0.38
CCNB2 O95067 1/20 0.37
CDK1 P06493 1/20 0.37
CCNB1 P14635 1/20 0.37
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
CCNB3 Q8WWL7 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4051241 0.95 PI4KA (0.45) PI4KAPI4K2BPI4K2API4KBGPR84
SCHEMBL4052252 0.87 KDM4C (0.41) PI4KAPI4K2BPI4K2API4KBCCNB2
SCHEMBL4053122 0.80 GPR84 (0.47) PI4KAPI4K2BPI4K2API4KBGPR84
SCHEMBL4046994 0.80 ADORA1 (0.42) CDK1CCNB1GSK3AGSK3B
SCHEMBL4044144 0.77 METAP2 (0.34) PI4KAPI4K2BPI4K2API4KBHCAR2
SCHEMBL4042151 0.76 AAK1 (0.40) GPR84
SCHEMBL246326 0.76 PDE5A (0.53) PI4KAPI4K2BPI4K2API4KBHCAR2
SCHEMBL4047518 0.76 METAP2 (0.33) PI4KAPI4K2BPI4K2API4KB
SCHEMBL9648738 0.74 PI4KA (0.57) PI4KAPI4K2BPI4K2API4KBGPR84
SCHEMBL9406720 0.73 PI4KA (0.56) PI4KAPI4K2BPI4K2API4KBGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed