SCHEMBL4042151

SCHEMBL4042151

CC(C)CCc1nc2nccnc2[nH]1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 5/20 0.40
METAP2 P50579 1/20 0.36
METAP1 P53582 1/20 0.36
GPR84 Q9NQS5 1/20 0.36
NOS1 P29475 5/20 0.33
NOS2 P35228 5/20 0.33
NOS3 P29474 3/20 0.33
CYP2C9 P11712 1/20 0.33
SYK P43405 1/20 0.32
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
MAPT P10636 2/20 0.31
ALOX15 P16050 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HRH4 Q9H3N8 1/20 0.31
ESR1 P03372 2/20 0.31
ESR2 Q92731 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4053122 0.90 GPR84 (0.47) AAK1METAP2METAP1GPR84NOS1
SCHEMBL4047518 0.85 METAP2 (0.33) AAK1METAP2METAP1
SCHEMBL4053441 0.82 ADORA3 (0.40) METAP2METAP1PDE3BPDE3AMAPT
SCHEMBL4052252 0.80 KDM4C (0.41) METAP2METAP1NOS1NOS2NOS3
SCHEMBL4051241 0.77 PI4KA (0.45) GPR84
SCHEMBL4046923 0.76 PI4KA (0.51) GPR84
SCHEMBL4046994 0.76 ADORA1 (0.42) METAP2METAP1HTTSMN1; SMN2
SCHEMBL4044137 0.75 PDE9A (0.38) METAP2METAP1
SCHEMBL4047123 0.72 METAP2 (0.36) METAP2METAP1
SCHEMBL4052403 0.72 METAP2 (0.36) METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009029592-A1 HETEROBICYCLIC-SUBSTITUTED QUINOLONES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS KALYPSYS, INC. (US) 2009-03-05 WO disclosed