SCHEMBL4047173

SCHEMBL4047173

CCCC(NC(=O)Oc1ccoc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 2/20 0.35
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
ALDH1A1 P00352 2/20 0.33
CYP1A2 P05177 1/20 0.33
FKBP1A P62942 1/20 0.33
TSHR P16473 1/20 0.33
GPR132 Q9UNW8 3/20 0.32
PREP P48147 1/20 0.32
FAP Q12884 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4049268 0.93 SMYD3 (0.35) SMYD3CYP2C9CYP2C19ALDH1A1FKBP1A
SCHEMBL4048306 0.93 CTSK (0.38) SMYD3ALDH1A1
SCHEMBL4044048 0.90 HSD17B10 (0.37) SMYD3ALDH1A1TSHRPREPFAP
SCHEMBL4047756 0.89 CTSL (0.38) FKBP1AGPR132
SCHEMBL4043998 0.89 FKBP1A (0.37) SMYD3FKBP1A
SCHEMBL4051063 0.88 SMYD3 (0.36) SMYD3CYP2C9CYP2C19ALDH1A1CYP1A2
SCHEMBL4047844 0.88 SMYD3 (0.35) SMYD3FKBP1A
SCHEMBL4045208 0.88 SMYD3 (0.35) SMYD3CYP2C9CYP2C19ALDH1A1CYP1A2
SCHEMBL4051473 0.88 CTSK (0.34) ALDH1A1GPR132PREPFAP
SCHEMBL4047765 0.87 PREP (0.35) ALDH1A1PREPFAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed
US-20060100431-A1 Biologically active compounds AMURA THERAPEUTICS LIMITED (GB) 2006-05-11 US claimed
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP disclosed
US-20060100431-A1 Biologically active compounds AMURA THERAPEUTICS LIMITED (GB) 2006-05-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060100431-A1 Biologically active compounds SOST, CTSK, CTSS SMYD3 4011/4885CYP2C9 80/4885CYP2C19 430/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.