SCHEMBL4047831

SCHEMBL4047831

CCCC(NC(=O)Oc1ccsc1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1ccccn1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PREP P48147 2/20 0.35
FAP Q12884 2/20 0.35
ELANE P08246 1/20 0.34
CTSK P43235 3/20 0.33
KMT2A Q03164 1/20 0.31
GAA P10253 1/20 0.31
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045469 0.93 ELANE (0.37) ELANECTSKKMT2AGAAALDH1A1
SCHEMBL4043147 0.92 CTSK (0.40) ELANECTSKKMT2AALDH1A1
SCHEMBL4043139 0.90 ELANE (0.37) PREPFAPELANECTSKKMT2A
SCHEMBL4046503 0.90 CTSL (0.37) PREPFAPCTSK
SCHEMBL4045653 0.89 CTSS (0.38) ELANECTSKKMT2A
SCHEMBL4038257 0.89 PREP (0.34) PREPFAPELANECTSKKMT2A
SCHEMBL4045026 0.88 CTSK (0.36) PREPFAPELANECTSKGAA
SCHEMBL4044691 0.88 PREP (0.35) PREPFAPELANECTSK
SCHEMBL4047765 0.88 PREP (0.35) PREPFAPELANECTSKKMT2A
SCHEMBL4045208 0.87 SMYD3 (0.35) PREPFAPALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed
EP-1463728-B1 FUSED CYCLIC MODULATORS OF NUCLEAR HORMONE RECEPTOR FUNCTION BRISTOL MYERS SQUIBB CO (US) 2009-01-14 EP disclosed