SCHEMBL4048801

SCHEMBL4048801

CCCC(NC(=O)Oc1cc2cccc(OC)c2o1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)c1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 17/20 0.39
CTSL P07711 17/20 0.39
CTSS P25774 13/20 0.39
CTSB P07858 3/20 0.39
CTSV O60911 2/20 0.39
ALDH1A1 P00352 2/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
HPGD P15428 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4045839 0.93 CTSK (0.45) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4045167 0.91 ALDH1A1 (0.38) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL4047709 0.91 ALDH1A1 (0.34) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4044711 0.90 CTSK (0.47) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4042524 0.88 CHRNA7 (0.37) ALDH1A1KDM4ENPC1HPGD
SCHEMBL4042533 0.87 CTSK (0.40) CTSKCTSLCTSSCTSBCTSV
SCHEMBL4051523 0.87 ALDH1A1 (0.37) CTSKCTSLCTSSALDH1A1KDM4E
SCHEMBL4046844 0.86 HPGD (0.32) CTSKALDH1A1KDM4EHPGDRAB9A
SCHEMBL4045579 0.86 HPGD (0.32) ALDH1A1KDM4ENPC1HPGDRAB9A
SCHEMBL4039150 0.85 CHRNA7 (0.36) CTSKCTSSALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed