SCHEMBL4049254

SCHEMBL4049254

CCCC(NC(=O)Oc1cc2cc(OC)ccc2o1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.40
CHRNA7 P36544 1/20 0.40
CHRNA4 P43681 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
KMT2A Q03164 1/20 0.35
PTAFR P25105 6/20 0.35
TAS1R3 Q7RTX0 4/20 0.35
TAS1R1 Q7RTX1 4/20 0.35
SMYD3 Q9H7B4 2/20 0.34
KCNA5 P22460 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4046703 0.93 CHRNB2 (0.42) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4049417 0.93 CHRNB2 (0.40) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4046863 0.92 SMYD3 (0.35) CHRNB2CHRNA7CHRNA4SMYD3
SCHEMBL4043869 0.91 KCNQ1 (0.37) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4046322 0.90 CHRNB2 (0.38) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4047814 0.89 CHRNB2 (0.36) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4048091 0.89 HPGD (0.38) ALDH1A1HPGDTAS1R3TAS1R1
SCHEMBL4044034 0.88 CHRNB2 (0.41) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4043632 0.88 CHRNA7 (0.40) CHRNB2CHRNA7CHRNA4ALDH1A1KMT2A
SCHEMBL4047844 0.87 SMYD3 (0.35) SMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed