SCHEMBL4046322

SCHEMBL4046322

COc1ccc2oc(OC(=O)NC(Cc3cccs3)C(=O)N3CCC4C3C(=O)CN4S(=O)(=O)Cc3cccnc3)cc2c1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.38
CHRNA7 P36544 1/20 0.38
CHRNA4 P43681 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
TRPM8 Q7Z2W7 2/20 0.34
KMT2A Q03164 1/20 0.32
SMYD3 Q9H7B4 2/20 0.32
F12 P00748 1/20 0.32
USP30 Q70CQ3 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
TAS1R3 Q7RTX0 2/20 0.31
TAS1R1 Q7RTX1 2/20 0.31
CTSB P07858 1/20 0.31
CTSS P25774 1/20 0.31
CTSK P43235 1/20 0.31
KCNQ1 P51787 1/20 0.31
PTAFR P25105 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4043432 0.91 KCNQ1 (0.38) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4046703 0.91 CHRNB2 (0.42) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4049254 0.90 CHRNB2 (0.40) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4049417 0.90 CHRNB2 (0.40) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4045350 0.90 CHRNB2 (0.34) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4051635 0.89 HPGD (0.37) ALDH1A1HPGDTRPM8USP30CTSB
SCHEMBL4044847 0.89 CHRNB2 (0.39) CHRNB2CHRNA7CHRNA4ALDH1A1HPGD
SCHEMBL4049501 0.86 CTSK (0.40) HPGDTRPM8CTSBCTSSCTSK
SCHEMBL4038978 0.85 USP30 (0.34) HPGDTRPM8USP30CTSBCTSS
SCHEMBL4044402 0.84 GAA (0.36) ALDH1A1TRPM8USP30TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed