SCHEMBL4050147

SCHEMBL4050147

CC(C)CC(NC(=O)Oc1ccc2ccccc2c1)C(=O)N1CCC2C1C(=O)CN2S(=O)(=O)Cc1cccnc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSK P43235 8/20 0.40
MMP1 P03956 2/20 0.37
MMP3 P08254 2/20 0.37
MMP9 P14780 2/20 0.37
CTSL P07711 4/20 0.36
CTSS P25774 3/20 0.36
CTSB P07858 2/20 0.36
SMYD3 Q9H7B4 2/20 0.36
FKBP1A P62942 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4041373 0.93 CTSK (0.38) CTSKMMP1MMP3MMP9CTSL
SCHEMBL4047844 0.93 SMYD3 (0.35) CTSKSMYD3FKBP1A
SCHEMBL4043952 0.92 CTSK (0.42) CTSKCTSLCTSSCTSBFKBP1A
SCHEMBL4040677 0.90 CTSK (0.41) CTSKMMP1MMP3MMP9CTSL
SCHEMBL4050939 0.89 CTSK (0.37) CTSKCTSLCTSSCTSBSMYD3
SCHEMBL4042904 0.89 CTSK (0.39) CTSKMMP1MMP3MMP9CTSL
SCHEMBL4051166 0.89 CTSK (0.39) CTSKMMP1MMP3MMP9CTSL
SCHEMBL4040754 0.88 CTSK (0.40) CTSKCTSLCTSSCTSB
SCHEMBL4048306 0.88 CTSK (0.38) CTSKCTSLCTSSCTSBSMYD3
SCHEMBL4042764 0.88 CTSK (0.38) CTSKCTSLCTSSCTSBSMYD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1546150-B1 PYRROLE DERIVATIVES AS INHIBITORS OF CYTEINE PROTEASES AMURA THERAPEUTICS LTD (GB) 2009-03-04 EP claimed