SCHEMBL40537

SCHEMBL40537

O=C1CC(c2ccc(Cl)cc2Cl)=NO1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.60
CRBN Q96SW2 1/20 0.45
PDCD1 Q15116 1/20 0.43
CD274 Q9NZQ7 1/20 0.43
NPSR1 Q6W5P4 3/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39
POLB P06746 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2C19 P33261 2/20 0.39
LMNA P02545 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
MCL1 Q07820 1/20 0.39
HKDC1 Q2TB90 1/20 0.39
AHR P35869 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2917568 0.84 NOTUM (0.57) NOTUMALDH1A1HPGDKMT2ALMNA
SCHEMBL9782150 0.75 NOTUM (1.00) NOTUMPDCD1CD274NPSR1ALDH1A1
SCHEMBL7582370 0.70 AXL (0.46) CRBNPDCD1CD274ALDH1A1HPGD
SCHEMBL29624840 0.66 AHR (0.64) ALDH1A1CYP3A4MAPTAHRHSD11B1
SCHEMBL464507 0.66 AHR (0.64) ALDH1A1CYP3A4MAPTAHRHSD11B1
SCHEMBL19872979 0.66 KIF11 (0.40) CRBNNPSR1ALDH1A1HPGDMEN1
SCHEMBL11571230 0.66 SMN1; SMN2 (0.47) CRBNPDCD1CD274ALDH1A1HPGD
SCHEMBL10389746 0.65 HPGD (0.57) HPGDPOLBMEN1KMT2ALMNA
SCHEMBL17085927 0.64 CRBN (0.40) CRBNPDCD1CD274NPSR1ALDH1A1
SCHEMBL181974 0.63 NOTUM (0.67) NOTUMPDCD1CD274ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120100989-A1 3-Aryl-4-(2-thienylmethylene)isoxazol-5(4H)-ones as Fungicides BAYER CROPSCIENCE AG (DE) 2012-04-26 US disclosed
WO-2011161035-A1 3-ARYL-4-(2-THIENYLMETHYLENE)-ISOXAZOL-5(4H)-ONES AS FUNGICIDES BAYER CROPSCIENCE AG (DE) 2011-12-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120100989-A1 3-Aryl-4-(2-thienylmethylene)isoxazol-5(4H)-ones as Fungicides CYP4X1, CYP4Z1, TH NOTUM 1620/4885CRBN 149/4885PDCD1 1223/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.