SCHEMBL4054074

SCHEMBL4054074

CC(=O)Oc1ccccc1-c1cc2ccccc2s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 5/20 0.43
MAOB P27338 1/20 0.43
APP P05067 1/20 0.43
ERN1 O75460 1/20 0.42
ADORA2A P29274 2/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA1 P30542 1/20 0.42
TSHR P16473 3/20 0.41
KDM4E B2RXH2 2/20 0.41
HSD17B10 Q99714 2/20 0.41
TMIGD3 P0DMS9 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ESR1 P03372 1/20 0.41
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
HMGB1 P09429 1/20 0.41
HPGD P15428 1/20 0.41
GGT1 P19440 1/20 0.41
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17167476 0.80 APP (0.59) TNFRSF1AAPPERN1KDM4EALDH1A1
SCHEMBL7639250 0.77 APP (0.58) TNFRSF1AAPPERN1TSHRHSD17B10
SCHEMBL4851399 0.76 BCL2L1 (0.50) PTGS2BCL2L1LMNACYP1A2GAA
SCHEMBL19133572 0.75 APP (0.57) APPERN1BCL2L1
SCHEMBL8676653 0.75 PTGS2 (0.61) MAOBTSHRKDM4EHSD17B10ALDH1A1
SCHEMBL17367221 0.73 SLC6A3 (0.55) TNFRSF1AAPPERN1TSHRHSD17B10
SCHEMBL12854022 0.73 APP (0.55) APPERN1BCL2L1
SCHEMBL4048688 0.72 TMIGD3 (0.58) MAOBERN1ADORA2ATSHRKDM4E
SCHEMBL17799582 0.72 CA12 (0.58) APPERN1HSD17B10ALDH1A1BCL2L1
SCHEMBL25744524 0.71 APP (0.44) TNFRSF1AAPPERN1BCL2L1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024371-A1 PHENANTHRENE DERIVATIVES AS MPGES-1 INHIBITORS Merck Frosst Canada Ltd. (CA) 2009-02-18 EP disclosed
WO-2007134434-A1 PHENANTHRENE DERIVATIVES AS MPGES-1 INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-11-29 WO disclosed