SCHEMBL4055219

SCHEMBL4055219

CC(=O)Oc1ccc(Cl)cc1-c1ccsc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMIGD3 P0DMS9 2/20 0.53
ADORA2A P29274 2/20 0.53
CNR1 P21554 1/20 0.41
BACE1 P56817 1/20 0.40
SLC6A9 P48067 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.40
NR1H4 Q96RI1 1/20 0.39
CFD P00746 1/20 0.39
AMY1A P0DUB6 1/20 0.39
ABCB11 O95342 1/20 0.38
ALDH1A1 P00352 3/20 0.37
HPGD P15428 2/20 0.37
ALOX5 P09917 1/20 0.37
KMT2A Q03164 3/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
MAPT P10636 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MEN1 O00255 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3830673 0.86 CNR1 (0.41) TMIGD3ADORA2ACNR1SLC6A9PTGDR2
SCHEMBL5764049 0.82 BACE1 (0.54) BACE1PTGDR2NR1H4CFDAMY1A
SCHEMBL5572529 0.80 BACE1 (0.53) TMIGD3ADORA2ABACE1SLC6A9PTGDR2
SCHEMBL24574845 0.74 SLC6A9 (0.47) TMIGD3ADORA2ASLC6A9CFDKMT2A
SCHEMBL5763924 0.74 PTGDR2 (0.49) BACE1PTGDR2CFDAMY1AALDH1A1
SCHEMBL1690266 0.73 PTGDR2 (0.42) BACE1PTGDR2NR1H4CFDAMY1A
SCHEMBL11338058 0.72 KDM4E (0.58) NR1H4CFDAMY1AABCB11ALDH1A1
SCHEMBL28179635 0.72 CYP2A6 (0.42) CNR1KMT2ARAB9ANPC1MAPT
SCHEMBL3691064 0.72 KMT2A (0.61) NR1H4CFDABCB11ALDH1A1HPGD
SCHEMBL5004411 0.72 CNR1 (0.42) TMIGD3ADORA2ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2024371-A1 PHENANTHRENE DERIVATIVES AS MPGES-1 INHIBITORS Merck Frosst Canada Ltd. (CA) 2009-02-18 EP disclosed
WO-2007134434-A1 PHENANTHRENE DERIVATIVES AS MPGES-1 INHIBITORS MERCK FROSST CANADA LTD. (CA) 2007-11-29 WO disclosed