SCHEMBL4055238

SCHEMBL4055238

O=[PH](O)OCc1ccc(F)cc1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.48
AGXT P21549 2/20 0.48
MAOB P27338 7/20 0.44
APP P05067 1/20 0.44
NR4A2 P43354 2/20 0.43
PARP10 Q53GL7 1/20 0.42
TAAR1 Q96RJ0 1/20 0.40
CTBP2 P56545 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA7 P43166 1/20 0.39
CA9 Q16790 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Butane SCHEMBL6056712 0.93 IDO1 (0.42) IDO1AGXTMAOBAPPNR4A2
SCHEMBL22589820 0.83 IDO1 (0.48) IDO1APPTAAR1CA2
SCHEMBL4055235 0.83 IDO1 (0.52) IDO1AGXTMAOBAPPNR4A2
SCHEMBL17061043 0.81 CYP3A4 (0.50) IDO1APP
SCHEMBL4076437 0.81 APP (0.46) IDO1MAOBAPPCA2CA9
SCHEMBL3365610 0.81 PRSS1 (0.39) IDO1APPCA12CA1CA2
SCHEMBL6020751 0.79 IDO1 (0.31) IDO1APPCA2CA9
SCHEMBL4938371 0.79 IDO1 (0.48) IDO1MAOBAPPTAAR1CA12
SCHEMBL5432095 0.79 AGXT (0.48) IDO1AGXTMAOBPARP10TAAR1
SCHEMBL4066062 0.79 CES2 (0.38) IDO1APPCA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020219718-A1 SMALL MOLECULE AUTOPHAGY INDUCERS FOR THE TREATMENT OF CANCER AND NEURODEGENERATIVE DISEASES JOHN WAYNE CANCER INSTITUTE (US) 2020-10-29 WO disclosed
CN-111801333-A 10- (di (phenyl) methyl) -4-hydroxy-8, 9,9a, 10-tetrahydro-7H-pyrrolo [1',2':4,5] pyrazino [1,2-b ] pyridazine-3, 5-dione derivatives and related compounds as inhibitors of orthomyxovirus replication for the treatment of influenza 诺华股份有限公司 2020-10-20 CN disclosed
CN-107078352-B Nonaqueous electrolyte solution and nonaqueous electrolyte secondary battery using same 三菱化学株式会社 2020-04-28 CN disclosed
WO-2009119880-A1 SUBSTITUTED PYRAZOLE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-01 WO disclosed