SCHEMBL4055235

SCHEMBL4055235

O=[PH](OCc1ccc(F)cc1)OCc1ccc(F)cc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 5/20 0.52
AGXT P21549 2/20 0.52
MAOB P27338 7/20 0.47
TAAR1 Q96RJ0 1/20 0.43
APP P05067 1/20 0.42
NR4A2 P43354 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
PARP10 Q53GL7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4055238 0.83 IDO1 (0.48) IDO1AGXTMAOBTAAR1APP
SCHEMBL11249728 0.79 IDO1 (0.41) IDO1AGXTMAOBAPPNR4A2
SCHEMBL8855401 0.79 IDO1 (0.50) IDO1TAAR1APPCA2
SCHEMBL742829 0.79 ALDH1A1 (0.46) MAOBAPPLOXL2CA2CA9
SCHEMBL17061042 0.77 CYP3A4 (0.52) IDO1APP
SCHEMBL6020749 0.77 CA2 (0.32) CA2CA9
SCHEMBL17181662 0.77 IDO1 (0.52) IDO1AGXTMAOBTAAR1APP
SCHEMBL9849327 0.77 TRPA1 (0.39) IDO1CA2CA9
SCHEMBL5432093 0.77 AGXT (0.52) IDO1AGXTMAOBTAAR1CA1
SCHEMBL2016123 0.77 IDO1 (0.52) IDO1MAOBTAAR1APPCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020219718-A1 SMALL MOLECULE AUTOPHAGY INDUCERS FOR THE TREATMENT OF CANCER AND NEURODEGENERATIVE DISEASES JOHN WAYNE CANCER INSTITUTE (US) 2020-10-29 WO disclosed
CN-111801333-A 10- (di (phenyl) methyl) -4-hydroxy-8, 9,9a, 10-tetrahydro-7H-pyrrolo [1',2':4,5] pyrazino [1,2-b ] pyridazine-3, 5-dione derivatives and related compounds as inhibitors of orthomyxovirus replication for the treatment of influenza 诺华股份有限公司 2020-10-20 CN disclosed
CN-107078352-B Nonaqueous electrolyte solution and nonaqueous electrolyte secondary battery using same 三菱化学株式会社 2020-04-28 CN disclosed
WO-2009119880-A1 SUBSTITUTED PYRAZOLE DERIVATIVES AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-10-01 WO disclosed