SCHEMBL4055948

SCHEMBL4055948

COc1ccc(C2(C#N)CCc3nc(N)ncc3C2)c2c3cc([N+](=O)[O-])ccc3n(C)c12

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
BACE1 P56817 1/20 0.36
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 4/20 0.32
ALDH1A1 P00352 3/20 0.32
LMNA P02545 2/20 0.32
ROCK1 Q13464 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.31
HTT P42858 1/20 0.31
APP P05067 1/20 0.30
BCHE P06276 1/20 0.30
ACHE P22303 1/20 0.30
SCARB1 Q8WTV0 1/20 0.30
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050217 0.89 BACE1 (0.32) BACE1MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL4061738 0.88 HTR2A (0.31) ALDH1A1HTTHTR1ADRD2HTR2A
SCHEMBL4054950 0.85 KDM4E (0.32) MAPTALDH1A1HTT
SCHEMBL4050626 0.81 PDE4A (0.39) BACE1TDP1MAPTALDH1A1LMNA
SCHEMBL4052813 0.80 KDM4E (0.31) ALDH1A1HTT
SCHEMBL4540659 0.76 KDM4E (0.32)
SCHEMBL4051064 0.75 ALDH1A1 (0.34) KMT2AMAPTALDH1A1SMN1; SMN2HTT
SCHEMBL4060742 0.73 HSD17B10 (0.32) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL4053970 0.72 KDM4E (0.31)
SCHEMBL4059118 0.72 CYP17A1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO claimed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed