SCHEMBL4050217

SCHEMBL4050217

COc1ccc(C2(C#N)CCc3ncncc3C2)c2c3cc([N+](=O)[O-])ccc3n(C)c12

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.32
ALDH1A1 P00352 4/20 0.32
MAPT P10636 3/20 0.32
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
HTR1A P08908 1/20 0.30
DRD2 P14416 1/20 0.30
DRD1 P21728 1/20 0.30
HTR2A P28223 1/20 0.30
HPGD P15428 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
F2RL3 Q96RI0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4055948 0.89 MEN1 (0.37) BACE1ALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL4540659 0.87 KDM4E (0.32)
SCHEMBL4060742 0.85 HSD17B10 (0.32) ALDH1A1MAPTHPGD
SCHEMBL4050626 0.82 PDE4A (0.39) BACE1ALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL4061738 0.76 HTR2A (0.31) ALDH1A1HTR1ADRD2HTR2AHPGD
SCHEMBL4051064 0.75 ALDH1A1 (0.34) ALDH1A1MAPTSMN1; SMN2HTR1ADRD2
SCHEMBL4059123 0.75
SCHEMBL4053970 0.73 KDM4E (0.31)
SCHEMBL13693578 0.72 PIN1 (0.31)
SCHEMBL4062215 0.70 KDR (0.34) ALDH1A1MAPTSMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO claimed
WO-2009115874-A2 NOVEL HETEROCYCLIC COMPOUNDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION MATRIX LABORATORIES LTD. (IN) 2009-09-24 WO disclosed