SCHEMBL4057654

SCHEMBL4057654

CS(=O)(=O)OCc1ccc2sccc2c1

nearest known ligand 0.51

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.51
CA2 P00918 10/20 0.51
CA12 O43570 7/20 0.51
PDE10A Q9Y233 1/20 0.42
MRGPRX4 Q96LA9 1/20 0.41
SIGMAR1 Q99720 1/20 0.39
PTPRC P08575 1/20 0.37
PTPN6 P29350 1/20 0.37
PTPN11 Q06124 1/20 0.37
PTPN22 Q9Y2R2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL48794 0.80 SIGMAR1 (0.53) CYP2A6CA2CA12PDE10ASIGMAR1
SCHEMBL48037 0.78 SIGMAR1 (0.57) CYP2A6CA2CA12PDE10ASIGMAR1
SCHEMBL3144878 0.78 CYP2A6 (0.59) CYP2A6CA2CA12PDE10AMRGPRX4
SCHEMBL28707496 0.75 CYP2A6 (0.51) CYP2A6CA2CA12PDE10A
SCHEMBL29469352 0.75 CYP2A6 (0.51) CYP2A6CA2CA12PDE10A
SCHEMBL5547137 0.74 CYP2A6 (0.54) CYP2A6CA2CA12PDE10AMRGPRX4
SCHEMBL2962869 0.73 CYP2A6 (0.53) CYP2A6CA2CA12PDE10AMRGPRX4
SCHEMBL4952656 0.73 CA2 (0.58) CA2CA12PTPN11
SCHEMBL25226263 0.73 CA2 (0.36) CA2SIGMAR1
SCHEMBL16727006 0.73 CYP2A6 (0.39) CYP2A6CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111501-A1 DERIVATIVES OF IMIDAZO [4, 5-D] PYRIDAZINE AND THEIR USE AS ANTI-VIRAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2009-09-11 WO disclosed
US-20090226398-A1 ANTI-VIRAL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE GENELABS TECHNOLOGIES, INC. 2009-09-10 US disclosed
US-20050209274-A1 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor ABOTT LABORATORIES 2005-09-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209274-A1 Antagonists of melanin concentrating hormone effects on the melanin concentrating hormone receptor MCHR1, MCHR2, MC1R CYP2A6 2701/4885CA2 2859/4885CA12 3894/4885
US-20090226398-A1 ANTI-VIRAL COMPOUNDS, COMPOSITIONS, AND METHODS OF USE MAVS, SARS1, HAVCR2 CYP2A6 947/4885CA2 1373/4885CA12 495/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.