SCHEMBL4060561

SCHEMBL4060561

NC(=O)Cc1nc2ncccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.51
KMT2A Q03164 1/20 0.46
HPSE Q9Y251 1/20 0.45
METAP1 P53582 2/20 0.44
ALDH1A1 P00352 2/20 0.44
CYP2C9 P11712 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
DAGLA Q9Y4D2 1/20 0.44
ATM Q13315 1/20 0.44
PDE5A O76074 2/20 0.43
METAP2 P50579 1/20 0.43
HPGD P15428 1/20 0.43
DRD4 P21917 1/20 0.42
ITK Q08881 1/20 0.42
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3380916 0.79 HSD17B10 (0.65) NUDT1KMT2AALDH1A1CYP2C9NOS1
SCHEMBL3967813 0.78 NUDT1 (0.55) NUDT1KMT2AHPSEMETAP1CYP2C9
SCHEMBL4773954 0.78 NUDT1 (0.59) NUDT1METAP1ALDH1A1CYP2C9NOS1
SCHEMBL4347800 0.78 NUDT1 (0.55) NUDT1KMT2AHPSEMETAP1CYP2C9
SCHEMBL31587712 0.78 NUDT1 (0.55) NUDT1KMT2AHPSEMETAP1CYP2C9
SCHEMBL7002580 0.78 NUDT1 (0.58) NUDT1METAP1ALDH1A1CYP2C9NOS1
SCHEMBL29535177 0.77 CHRM1 (0.61) NUDT1KMT2ACYP2C9NOS1NOS2
SCHEMBL30943978 0.77 NUDT1 (0.58) NUDT1KMT2AHPSEMETAP1ALDH1A1
SCHEMBL853165 0.77 NUDT1 (0.58) NUDT1KMT2AHPSEMETAP1ALDH1A1
SCHEMBL2207637 0.76 MAPT (0.63) ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575952-B1 SYNTHESIS OF HETEROARYL ACETAMIDES MALLINCKRODT INC (US) 2009-02-18 EP claimed