SCHEMBL406134

SCHEMBL406134

CNC(=O)CCCCC(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 2/20 0.46
KDM4A O75164 1/20 0.46
PHF8 Q9UPP1 1/20 0.46
KDM2A Q9Y2K7 1/20 0.46
DEGS1 O15121 1/20 0.44
LMNA P02545 3/20 0.43
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
FAAH O00519 2/20 0.41
MAPK1 P28482 1/20 0.41
THRB P10828 1/20 0.39
CA1 P00915 2/20 0.39
BLM P54132 2/20 0.39
CYP1A2 P05177 1/20 0.39
POLB P06746 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
TSHR P16473 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10890772 0.98 KDM4C (0.49) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL24496288 0.98 KDM4C (0.49) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL12188679 0.98 KDM4C (0.49) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL23640057 0.98 KDM4C (0.49) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL10290720 0.98 KDM4C (0.49) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL13223739 0.93 LMNA (0.44) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL12299087 0.92 LMNA (0.48) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL1709869 0.83
SCHEMBL9437025 0.83 LMNA (0.40) KDM4CKDM4APHF8KDM2ADEGS1
SCHEMBL7753090 0.83 LMNA (0.57) LMNAMEN1KMT2AFAAHMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11834458-B2 Anti-cancer nuclear hormone receptor-targeting compounds NUVATION BIO INC. (US) 2023-12-05 US disclosed
US-11826430-B2 Anti-cancer nuclear hormone receptor-targeting compounds NUVATION BIO INC. (US) 2023-11-28 US disclosed
EP-4223309-A1 COMBINATION THERAPY WITH CONTROLLED-RELEASE CNP AGONISTS Ascendis Pharma Growth Disorders A/S (DK) 2023-08-09 EP disclosed
EP-3518930-B1 COMBINATION THERAPY WITH CONTROLLED-RELEASE CNP AGONISTS ASCENDIS PHARMA GROWTH DISORDERS AS (DK) 2023-03-08 EP disclosed
WO-2023283831-A1 VIRUS MAIN PROTEASE INHIBITOR, PREPARATION METHOD THEREFOR, AND USE 上海药明康德新药开发有限公司 2023-01-19 WO disclosed
US-20220218829-A1 NUCLEIC ACID CONJUGATES AND USES THEREOF TRANSLATE BIO MA, INC. (US) 2022-07-14 US disclosed
US-20210214316-A1 ANTI-CANCER NUCLEAR HORMONE RECEPTOR-TARGETING COMPOUNDS SAGARD HOLDINGS MANAGER LP, AS ADMINISTRATIVE AGENT (CA) 2021-07-15 US disclosed
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2021097046-A1 ANTI-CANCER NUCLEAR HORMONE RECEPTOR-TARGETING COMPOUNDS NUVATION BIO INC. (US) 2021-05-20 WO disclosed
US-20200360523-A1 ANTI-CANCER NUCLEAR HORMONE RECEPTOR-TARGETING COMPOUNDS SAGARD HOLDINGS MANAGER LP, AS ADMINISTRATIVE AGENT (CA) 2020-11-19 US disclosed
US-20120064002-A1 Enantiomer-pure (4S,8S)- and (4R,8R)-4-p-Nitrobenzyl-8-methyl-3,6,9-triaza-3N,6N,9N-tricarboxymethyl-1,11-undecanedioic Acid and Derivatives Thereof, Process for their Production and Use for the Production of Pharmaceutical Agents LEHMANN LUTZ (DE) 2012-03-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210214316-A1 ANTI-CANCER NUCLEAR HORMONE RECEPTOR-TARGETING COMPOUNDS NCOA1, NCOR1, NCOA3 KDM4C 2613/4885KDM4A 1999/4885PHF8 1968/4885
US-20200360523-A1 ANTI-CANCER NUCLEAR HORMONE RECEPTOR-TARGETING COMPOUNDS NCOA1, NCOR1, NCOA3 KDM4C 2613/4885KDM4A 1999/4885PHF8 1968/4885
US-11834458-B2 Anti-cancer nuclear hormone receptor-targeting compounds NCOA1, NCOR1, NCOA3 KDM4C 2613/4885KDM4A 1999/4885PHF8 1968/4885
US-20120064002-A1 Enantiomer-pure (4S,8S)- and (4R,8R)-4-p-Nitrobenzyl-8-methyl-3,6,9-triaza-3N,6N,9N-tricarboxymethyl-1,11-undecanedioic Acid and Derivatives Thereof, Process for their Production and Use for the Production of Pharmaceutical Agents CYP4B1, CYP2B6, UGT2B7 KDM4C 1225/4885KDM4A 1165/4885PHF8 2201/4885
US-20220218829-A1 NUCLEIC ACID CONJUGATES AND USES THEREOF FOLR1, SLC19A1, FOLR2 KDM4C 3225/4885KDM4A 3986/4885PHF8 2723/4885
US-11826430-B2 Anti-cancer nuclear hormone receptor-targeting compounds NCOA1, NCOR1, NCOA3 KDM4C 2613/4885KDM4A 1999/4885PHF8 1968/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.