SCHEMBL4065260

SCHEMBL4065260

COC(=O)Oc1cc(C)c2[nH]c(=O)[nH]c2c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.37
MAPT P10636 4/20 0.37
GAA P10253 2/20 0.37
GLA P06280 1/20 0.36
CYP1A2 P05177 1/20 0.36
PDE3B Q13370 4/20 0.35
PDE3A Q14432 4/20 0.35
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
HSD17B10 Q99714 2/20 0.35
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
ALDH1A1 P00352 4/20 0.33
BCL6 P41182 1/20 0.33
BCOR Q6W2J9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3965692 0.84 KDM4E (0.41) KDM4EMAPTGAAGLAPDE3B
SCHEMBL2491701 0.75 CREBBP (0.40) KDM4EMAPTGAAGLAHSD17B10
SCHEMBL13907978 0.74 BCL6 (0.45) KDM4EMAPTGAACYP1A2HSD17B10
SCHEMBL3963475 0.73 ALDH1A1 (0.40) ALDH1A1HPGD
SCHEMBL9237989 0.71 KMT2A (0.42) KDM4EMAPTGAAHSD17B10MTNR1A
SCHEMBL13907960 0.68 TPMT (0.42) KDM4EMAPTGAAGRIN2DGRIN3B
SCHEMBL2257694 0.68 GRIN2D (0.69) KDM4EMAPTGAAPDE3BPDE3A
SCHEMBL8426699 0.68 MEN1 (0.49) KDM4EMAPTHSD17B10ALDH1A1MAPK1
SCHEMBL8425770 0.67 TDP1 (0.55) KDM4EMAPTGAAALDH1A1RAB9A
SCHEMBL4240634 0.67 MAPT (0.39) KDM4EMAPTALDH1A1RAB9AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009034029-A2 1-SUBSTITUTED 4-HETEROCYCLYLPIPERIDINES FOR USE AS CGRP ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-03-19 WO disclosed