SCHEMBL4065892

SCHEMBL4065892

CC(C)(Cc1ccncc1C=O)NC(=O)O

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FTO Q9C0B1 3/20 0.36
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
SRC P12931 1/20 0.33
KDM6B O15054 2/20 0.33
ALKBH2 Q6NS38 1/20 0.33
ALKBH3 Q96Q83 1/20 0.33
KDM5B Q9UGL1 1/20 0.33
KDM2A Q9Y2K7 1/20 0.33
KDM3A Q9Y4C1 1/20 0.33
SSTR4 P31391 2/20 0.32
KDM4C Q9H3R0 5/20 0.32
RAB9A P51151 1/20 0.32
LATS1 O95835 2/20 0.32
TBXAS1 P24557 2/20 0.32
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072495 0.89 CYP2C9 (0.35) FTOALDH1A1CYP3A4CYP2C9CYP2C19
SCHEMBL1932047 0.72 RAB9A (0.49) ALDH1A1CYP3A4CYP2C9CYP2C19RAB9A
SCHEMBL31068616 0.71 CYP2A6 (0.42) CYP3A4CYP2C9CYP2C19
SCHEMBL14872350 0.71 CYP2A6 (0.42) CYP3A4CYP2C9CYP2C19
SCHEMBL4066043 0.71 NAPRT (0.51) ALDH1A1CYP3A4CYP2C9CYP2C19TBXAS1
SCHEMBL4606675 0.69 KDM4E (0.40) ALDH1A1RAB9AKDM4EMAPT
SCHEMBL27495542 0.69 CA12 (0.44) ALDH1A1CYP3A4CYP2C9CYP2C19SRC
SCHEMBL29951676 0.67 CYP2E1 (0.44) CYP3A4CYP2C9CYP2C19KDM4C
SCHEMBL29958096 0.67 AOC1 (0.35) CYP2C19
SCHEMBL13387995 0.66 KDM4C (0.39) ALDH1A1KDM6BKDM4CRAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1751155-B1 SUBSTITUTED AZACHINAZOLINES HAVING AN ANTIVIRAL ACTION BAYER HEALTHCARE AG (DE) 2009-01-07 EP disclosed
EP-1751155-A1 SUBSTITUTED AZACHINAZOLINES HAVING AN ANTIVIRAL ACTION Bayer HealthCare AG (DE) 2007-02-14 EP disclosed
WO-2005113552-A1 SUBSTITUTED AZACHINAZOLINES HAVING AN ANTIVIRAL ACTION BAYER HEALTHCARE AG (DE) 2005-12-01 WO disclosed