SCHEMBL4066152

SCHEMBL4066152

O=C(O)Cc1cc2c(Cl)c(Cl)ccc2[nH]c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MAPT P10636 4/20 0.44
KDM4E B2RXH2 4/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 1/20 0.44
GRIN2D O15399 3/20 0.43
GRIN3B O60391 3/20 0.43
GRIN1 Q05586 3/20 0.43
GRIN2A Q12879 3/20 0.43
GRIN2B Q13224 3/20 0.43
GRIN2C Q14957 3/20 0.43
GRIN3A Q8TCU5 3/20 0.43
PIM1 P11309 1/20 0.43
DAO P14920 1/20 0.42
GAA P10253 1/20 0.41
HRH4 Q9H3N8 1/20 0.41
GRIK1 P39086 1/20 0.40
GRIA1 P42261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4066394 0.78 PIM1 (0.50) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL31145982 0.77 GRIN2D (0.41) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL31145902 0.77 TSHR (0.44) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL4064969 0.74 HSD17B10 (0.46) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL8545427 0.73 RHEB (0.53) ALDH1A1KDM4EHPGDHSD17B10HRH4
SCHEMBL31146056 0.72 AKR1C2 (0.49) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL9756207 0.72 AKR1B1 (0.46) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL678203 0.71 DAO (0.49) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL708527 0.71 GRIN1 (0.57) ALDH1A1KDM4EMEN1KMT2AHPGD
SCHEMBL4900831 0.69 CXCL8 (0.50) CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049118-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SmithKline Beecham Corporation (US) 2009-04-22 EP disclosed
WO-2008011551-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-24 WO disclosed