SCHEMBL4064969

SCHEMBL4064969

O=C(O)Cc1cc2cc(Cl)c(Cl)cc2[nH]c1=O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 7/20 0.46
GRIN2D O15399 6/20 0.46
GRIN3B O60391 6/20 0.46
GRIN1 Q05586 6/20 0.46
GRIN2A Q12879 6/20 0.46
GRIN2B Q13224 6/20 0.46
GRIN2C Q14957 6/20 0.46
GRIN3A Q8TCU5 6/20 0.46
KDM4E B2RXH2 5/20 0.46
TSHR P16473 5/20 0.46
GRIA1 P42261 3/20 0.46
GRIA2 P42262 3/20 0.46
GRIA3 P42263 3/20 0.46
GRIA4 P48058 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.46
LMNA P02545 2/20 0.46
CYP1A2 P05177 2/20 0.46
MAPT P10636 2/20 0.46
MEN1 O00255 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4067945 0.82 HSD17B10 (0.61) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3713838 0.81 GRIN2D (0.43) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL9270023 0.78 SIRT1 (0.47) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL5678790 0.75 MAPK1 (0.61) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL30434363 0.75 MAPK1 (0.61) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL31146173 0.75 DAO (0.58) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3713356 0.75 GRIN2D (0.44) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL14128774 0.75 GRIA1 (0.53) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL4066152 0.74 ALDH1A1 (0.44) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL3711310 0.74 HSD17B10 (0.38) HSD17B10GRIN2DGRIN3BGRIN1GRIN2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049118-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SmithKline Beecham Corporation (US) 2009-04-22 EP disclosed
WO-2008011551-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-24 WO disclosed