SCHEMBL4067336

SCHEMBL4067336

CCOC(=O)CN(C(=O)OCC)c1cc(Cl)c(Oc2ccc(OCC)c(CC)c2)c(Cl)c1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.35
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
THRB P10828 6/20 0.35
THRA P10827 4/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
RORC P51449 3/20 0.34
MTNR1A P48039 1/20 0.33
MTNR1B P49286 1/20 0.33
LMNA P02545 1/20 0.33
HTT P42858 1/20 0.33
PLA2G7 Q13093 1/20 0.33
MAPK1 P28482 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3213016 0.92 THRB (0.38) ALDH1A1KDM4EMEN1KMT2ATHRB
SCHEMBL3222209 0.85 THRB (0.36) ALDH1A1THRBTHRARORCMTNR1A
SCHEMBL3225634 0.84 ALDH1A1 (0.39) ALDH1A1KDM4EMEN1KMT2ATHRB
SCHEMBL3233002 0.83 RORC (0.55) THRBTHRARORC
SCHEMBL3226662 0.83 PPARG (0.41) ALDH1A1THRBTHRALMNAMAPT
SCHEMBL3224353 0.82 THRB (0.41) ALDH1A1KDM4EMEN1KMT2ATHRB
SCHEMBL3227188 0.82 THRB (0.46) ALDH1A1THRBTHRARORC
SCHEMBL3223228 0.81 THRB (0.36) ALDH1A1MEN1KMT2ATHRBTHRA
SCHEMBL3227779 0.81 TSHR (0.38) ALDH1A1MEN1KMT2ATHRBTHRA
SCHEMBL3219867 0.80 THRB (0.40) ALDH1A1KDM4EMEN1KMT2ATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2079678-A2 SELECTIVE TR-BETA 1 AGONIST Cadila Healthcare Limited (IN) 2009-07-22 EP disclosed
WO-2008062469-A2 SELECTIVE TR-BETA 1 AGONIST CADILA HEALTHCARE LIMITED (IN) 2008-05-29 WO disclosed