SCHEMBL4070398

SCHEMBL4070398

c1ccc(-c2cc(-c3ncco3)c3ccc(-c4csc5ncncc45)cc3n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.38
TSHR P16473 1/20 0.38
HSD17B10 Q99714 1/20 0.38
MCL1 Q07820 3/20 0.37
ALDH1A1 P00352 5/20 0.36
HPGD P15428 4/20 0.36
KDM4E B2RXH2 3/20 0.36
MAPT P10636 3/20 0.36
HPGDS O60760 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
RECQL P46063 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
POLB P06746 1/20 0.34
CAMKK1 Q8N5S9 1/20 0.34
CAMKK2 Q96RR4 1/20 0.34
ACACA Q13085 3/20 0.33
DHODH Q02127 2/20 0.33
LTA4H P09960 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3986474 0.83 KDR (0.54) MAPK1TSHRHSD17B10MCL1HPGD
SCHEMBL14964882 0.72 FGFR1 (0.53) MAPK1ALDH1A1HPGDKDM4EMAPT
SCHEMBL3979887 0.70 KDR (0.67) MCL1ALDH1A1HPGDKDM4EKMT2A
SCHEMBL3981493 0.69 KDR (0.50) MAPK1MCL1HPGDKDM4EKMT2A
SCHEMBL3978118 0.67 KDR (0.55) MCL1HPGDKDM4EKMT2APOLB
SCHEMBL28297480 0.67 ACACA (0.48) MAPK1TSHRHSD17B10MCL1ALDH1A1
SCHEMBL3977506 0.65 KDR (0.59) MCL1ALDH1A1HPGDKDM4EMEN1
SCHEMBL30700550 0.64 DHFR (0.41) ALDH1A1KDM4EMAPTKMT2ALMNA
SCHEMBL2367997 0.64 LMNA (0.49) ALDH1A1MAPTMEN1KMT2ALMNA
SCHEMBL2368915 0.64 SMN1; SMN2 (0.38) MAPK1TSHRHSD17B10ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2051982-A1 6,6-BICYCLIC RING SUBSTITUTED SULFUR CONTAINING HETEROBICYCLIC PROTEIN KINASE INHIBITORS OSI Pharmaceuticals, Inc. (US) 2009-04-29 EP disclosed
WO-2008018881-A1 6,6-BICYCLIC RING SUBSTITUTED SULFUR CONTAINING HETEROBICYCLIC PROTEIN KINASE INHIBITORS OSI PHARMACEUTICALS, INC. (US) 2008-02-14 WO disclosed