SCHEMBL4071987

SCHEMBL4071987

O=C1COc2ccc(OC(F)(F)F)cc2[N]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.37
PIM1 P11309 1/20 0.37
ABL1 P00519 5/20 0.36
CES1 P23141 1/20 0.36
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
SCN4A P35499 2/20 0.35
SCN5A Q14524 2/20 0.35
SCN9A Q15858 2/20 0.35
SCN2A Q99250 2/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
GMNN O75496 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL315498 0.71 MAPT (0.53) NPC1RAB9AUSP2SMN1; SMN2MAPK1
SCHEMBL704966 0.71 MMP12 (0.55) ABL1CES1LMNAPKMSMN1; SMN2
SCHEMBL6757684 0.68 KIF11 (0.50) PIM1CES1
SCHEMBL31560396 0.67 PTGS1 (0.49) PIM1PTGS1PTGS2TP53GAA
SCHEMBL12316591 0.66 GRM5 (0.45) CHRM5CES1PTGS1PTGS2SCN4A
SCHEMBL1208429 0.65 PTGS1 (0.56) PIM1PTGS1PTGS2TP53GAA
SCHEMBL3881419 0.65 MAOA (0.58) CES1LMNAGAAKCNH2GPR3
SCHEMBL2953372 0.64 HTT (0.62) USP2CYP1A2CYP3A4KCNH2
SCHEMBL14775775 0.63 PTGS1 (0.51) PIM1PTGS1PTGS2
SCHEMBL2054544 0.63 PTGS1 (0.42) CHRM5PTGS1PTGS2GPR3CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049118-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SmithKline Beecham Corporation (US) 2009-04-22 EP disclosed
WO-2008011551-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-24 WO disclosed