SCHEMBL4072987

SCHEMBL4072987

CC(C)(C)C(COC(N)=O)c1ccc(Br)cc1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
CYP2D6 P10635 2/20 0.42
PKM P14618 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
ALOX5 P09917 1/20 0.41
EPHX1 P07099 2/20 0.37
LMNA P02545 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
POLB P06746 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20425505 1.00 CYP1A2 (0.42) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL1937037 0.86 CYP1A2 (0.44) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL28432379 0.84 CYP1A2 (0.62) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL1936445 0.83 PPARG (0.43) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL1935051 0.83 ADRB2 (0.43) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL3468423 0.79 ALOX5 (0.47) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL29213688 0.79 ALOX5 (0.47) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL28989195 0.77 CYP1A2 (0.47) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1
SCHEMBL1935792 0.76 HRH3 (0.47) KDM4EALDH1A1MEN1KMT2A
SCHEMBL28617148 0.74 MAPT (0.37) CYP1A2SMN1; SMN2CYP2D6PKMNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049118-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SmithKline Beecham Corporation (US) 2009-04-22 EP disclosed
WO-2008011551-A1 MORPHOLINYL AND PYRROLIDINYL ANALOGS SMITHKLINE BEECHAM CORPORATION (US) 2008-01-24 WO disclosed