SCHEMBL4074083

SCHEMBL4074083

O=C(O)CCCC(=O)NCc1cc(Cl)ccc1Cl

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.52
ALDH1A1 P00352 4/20 0.51
POLB P06746 2/20 0.51
HTT P42858 1/20 0.50
P2RX7 Q99572 2/20 0.49
KMT2A Q03164 1/20 0.49
RAB9A P51151 1/20 0.48
TP53 P04637 1/20 0.46
HPGD P15428 2/20 0.46
TRPV1 Q8NER1 1/20 0.46
TSHR P16473 1/20 0.46
GAA P10253 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074085 0.94 HTT (0.55) ALDH1A1HTTP2RX7KMT2ATP53
SCHEMBL4246819 0.80 P2RX7 (0.54) SMN1; SMN2ALDH1A1POLBHTTP2RX7
SCHEMBL3557506 0.79 P2RX7 (0.53) ALDH1A1POLBP2RX7KMT2ARAB9A
SCHEMBL7934893 0.78 P2RX7 (0.53) ALDH1A1POLBP2RX7KMT2ARAB9A
SCHEMBL29594946 0.78 TRPV1 (0.72) SMN1; SMN2ALDH1A1KMT2ATP53HPGD
SCHEMBL4074090 0.77 P2RX7 (0.40) ALDH1A1HTTP2RX7KMT2ATP53
SCHEMBL4079697 0.77 SMN1; SMN2 (0.75) SMN1; SMN2ALDH1A1HTTKMT2ARAB9A
SCHEMBL7905467 0.76 F13A1 (0.53) ALDH1A1RAB9ATP53
SCHEMBL20672330 0.75 F13A1 (0.56)
SCHEMBL11867707 0.75 ALDH1A1 (0.58) ALDH1A1HTTP2RX7KMT2ARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds PKD1, DDC, DPYD SMN1; SMN2 1061/4885ALDH1A1 158/4885POLB 1568/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.