SCHEMBL4074085

SCHEMBL4074085

O=C(CCCC(=O)NCc1cc(Cl)ccc1Cl)NCc1cc(Cl)ccc1Cl

nearest known ligand 0.55

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.55
KMT2A Q03164 2/20 0.53
P2RX7 Q99572 2/20 0.53
ALDH1A1 P00352 3/20 0.50
HPGD P15428 2/20 0.50
TP53 P04637 1/20 0.50
TRPV1 Q8NER1 2/20 0.48
MEN1 O00255 1/20 0.48
ERCC1 P07992 2/20 0.47
ERCC4 Q92889 2/20 0.47
TSHR P16473 1/20 0.47
LMNA P02545 1/20 0.46
MAPT P10636 1/20 0.46
GAA P10253 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4074083 0.94 SMN1; SMN2 (0.52) HTTKMT2AP2RX7ALDH1A1HPGD
SCHEMBL4246819 0.85 P2RX7 (0.54) HTTKMT2AP2RX7ALDH1A1MEN1
SCHEMBL7934893 0.83 P2RX7 (0.53) KMT2AP2RX7ALDH1A1MEN1ERCC1
SCHEMBL4074090 0.82 P2RX7 (0.40) HTTKMT2AP2RX7ALDH1A1HPGD
SCHEMBL3557506 0.81 P2RX7 (0.53) KMT2AP2RX7ALDH1A1TP53MEN1
SCHEMBL11867707 0.80 ALDH1A1 (0.58) HTTKMT2AP2RX7ALDH1A1TP53
SCHEMBL5797584 0.79 P2RX7 (0.49) KMT2AP2RX7ALDH1A1MEN1ERCC1
SCHEMBL626586 0.79 CYP2C9 (0.58) KMT2AP2RX7ALDH1A1MEN1ERCC1
SCHEMBL6649593 0.78 HTT (0.69) HTTKMT2AP2RX7ALDH1A1HPGD
SCHEMBL18887625 0.77 LMNA (0.50) HTTKMT2AP2RX7ALDH1A1ERCC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds PKD1, DDC, DPYD HTT 422/4885KMT2A 3604/4885P2RX7 2220/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.