SCHEMBL4076358

SCHEMBL4076358

COC(=O)C(Cc1ccc(Cl)cc1)NC(=O)CCC(=O)NC1CCC(Cc2ccc(C)cc2)(N(C)C)CC1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 10/20 0.43
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
OXTR P30559 1/20 0.41
HDAC1 Q13547 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
NOS2 P35228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL209932 0.92 AVPR1A (0.44) AVPR1AOXTRKMT2A
SCHEMBL208694 0.88 AVPR1A (0.41) AVPR1AL3MBTL1OXTR
SCHEMBL207560 0.83 POLB (0.41) AVPR1AKMT2A
SCHEMBL4049886 0.82 MAPT (0.45) ATML3MBTL1HDAC1HDAC6KMT2A
SCHEMBL208300 0.81 LMNA (0.50) KMT2A
SCHEMBL206987 0.80 POLB (0.56) KMT2A
SCHEMBL4079453 0.80 LMNA (0.43) AVPR1AOXTR
SCHEMBL206402 0.80 ALDH1A1 (0.41) L3MBTL1HDAC1HDAC6KMT2A
SCHEMBL4084189 0.79 HRH3 (0.40) L3MBTL1HDAC1HDAC6KMT2A
SCHEMBL2983415 0.79 MEN1 (0.45) L3MBTL1HDAC1HDAC6KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP disclosed