SCHEMBL4084189

SCHEMBL4084189

Cc1ccc(CC2(N(C)C)CCC(NC(=O)CCC(=O)NC(C)C(=O)O)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.40
OPRM1 P35372 2/20 0.39
OPRL1 P41146 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
KDM4E B2RXH2 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
NCOR2 Q9Y618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4079453 0.91 LMNA (0.43) HRH3OPRM1OPRL1HPGD
SCHEMBL206402 0.88 ALDH1A1 (0.41) OPRM1OPRL1ALDH1A1HPGDRAB9A
SCHEMBL207622 0.86 HRH3 (0.45) HRH3OPRM1OPRL1ALDH1A1HPGD
SCHEMBL209932 0.84 AVPR1A (0.44) MEN1KMT2A
SCHEMBL4081016 0.83 EPHX2 (0.45) OPRM1OPRL1ALDH1A1HPGDL3MBTL1
SCHEMBL208694 0.83 AVPR1A (0.41) ALDH1A1HPGDL3MBTL1
SCHEMBL5162372 0.83 RAB9A (0.43) OPRM1OPRL1ALDH1A1HPGDRAB9A
SCHEMBL4080671 0.82 OPRM1 (0.37) OPRM1OPRL1ALDH1A1HPGDRAB9A
SCHEMBL4075032 0.82 HPGD (0.40) OPRM1OPRL1ALDH1A1HPGDRAB9A
SCHEMBL4048631 0.82 KMT2A (0.51) OPRM1OPRL1ALDH1A1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed