SCHEMBL4078294

SCHEMBL4078294

O=C(O)CCCC(=O)NC1CCN(Cc2c(Cl)cccc2Cl)C1

nearest known ligand 0.61

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 5/20 0.61
SIGMAR1 Q99720 4/20 0.58
CX3CR1 P49238 2/20 0.51
ALDH1A1 P00352 1/20 0.48
KMT2A Q03164 1/20 0.48
BACE1 P56817 1/20 0.47
DRD2 P14416 2/20 0.46
DRD4 P21917 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4072400 0.96 CCR2 (0.61) CCR2SIGMAR1CX3CR1ALDH1A1KMT2A
SCHEMBL249743 0.81 CX3CR1 (0.44) CCR2SIGMAR1CX3CR1ALDH1A1DRD2
SCHEMBL3177907 0.74 KDM4E (0.48) CCR2SIGMAR1CX3CR1ALDH1A1BACE1
SCHEMBL11576999 0.74 SIGMAR1 (0.65) CCR2SIGMAR1BACE1DRD2DRD4
SCHEMBL205373 0.74 CCR2 (0.47) CCR2SIGMAR1CX3CR1ALDH1A1DRD2
SCHEMBL4074069 0.73 MEN1 (0.60) ALDH1A1KMT2A
SCHEMBL4844836 0.72 CCR2 (0.71) CCR2SIGMAR1DRD2DRD4
SCHEMBL4847367 0.72 CCR2 (0.71) CCR2SIGMAR1DRD2DRD4
SCHEMBL28741993 0.71 SIGMAR1 (0.77) SIGMAR1
SCHEMBL2445773 0.71 CXCR4 (0.54) SIGMAR1ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745010-B1 SUBSTITUTED CYCLOHEXYL-1,4-DIAMINE DERIVATIVES GRUENENTHAL GMBH (DE) 2009-08-05 EP claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US claimed
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds GRUENENTHAL GMBH (DE) 2007-05-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070112007-A1 Cyclohexyl-1, 4-diamine compounds PKD1, DDC, DPYD CCR2 2965/4885SIGMAR1 3262/4885CX3CR1 4296/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.