SCHEMBL4079236

SCHEMBL4079236

COC(=O)c1ccc(CCNNC(=O)OC(C)(C)C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.50
CYP4F2 P78329 1/20 0.49
LOXL2 Q9Y4K0 1/20 0.46
ALDH1A1 P00352 2/20 0.46
HPGD P15428 2/20 0.46
HSD17B10 Q99714 2/20 0.46
TP53 P04637 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C9 P11712 1/20 0.46
ALOX15 P16050 1/20 0.46
ALOX12 P18054 1/20 0.46
CYP2C19 P33261 1/20 0.46
CKS1B P61024 1/20 0.46
SKP2 Q13309 1/20 0.46
HIF1A Q16665 1/20 0.46
MGLL Q99685 1/20 0.46
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA12 O43570 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2654355 0.88 CA12 (0.48) ALDH1A1HPGDCYP1A2CYP3A4CYP2C9
SCHEMBL5766581 0.86 CA1 (0.51) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL1936202 0.86 MGLL (0.55) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL30754110 0.84 NPC1 (0.47) CA1CA2HDAC1HDAC6NPC1
SCHEMBL20581863 0.83 HPGD (0.46) ALDH1A1HPGDCA1CA2LMNA
SCHEMBL7328495 0.82 CTSK (0.50) CA1CA12CA7CA14MAPT
SCHEMBL4465651 0.82 MGLL (0.51) CYP4A11CYP4F2LOXL2MGLLCA1
SCHEMBL1054945 0.82 CYP4A11 (0.58) CYP4A11CYP4F2LOXL2ALDH1A1HPGD
SCHEMBL4082188 0.81 MAPT (0.59) CA1CA2CA12CA9MAPT
SCHEMBL5983006 0.81 CYP4A11 (0.57) CYP4A11CYP4F2LOXL2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4565565-A1 1,2-SUBSTITUTED 3-OXOPYRAZOLIDINE DERIVATIVES AS PROSTAGLANDIN E2 RECEPTOR 4 (EP4) AGONISTS FOR THE TREATMENT OF GASTROINTESTINAL AND PULMONARY DISEASES Nxera Pharma UK Limited (GB) 2025-06-11 EP disclosed
WO-2024028601-A1 1,2-SUBSTITUTED 3-OXOPYRAZOLIDINE DERIVATIVES AS PROSTAGLANDIN E2 RECEPTOR 4 (EP4) AGONISTS FOR THE TREATMENT OF GASTROINTESTINAL AND PULMONARY DISEASES HEPTARES THERAPEUTICS LIMITED (GB) 2024-02-08 WO disclosed
EP-1847533-B1 SIX-MEMBERED HETEROCYCLIC COMPOUND AND THE USE THEREOF ASAHI KASEI PHARMA CORP (JP) 2013-08-14 EP disclosed
US-7863312-B2 Pyrazolidinone compounds as ligands of the prostaglandin EP2 and/or EP4 receptors MERCK SERONO SA (CH) 2011-01-04 US disclosed
US-7531533-B2 6-Membered heterocyclic compound and use thereof ASAHI KASEI PHARMA CORPORATION (JP) 2009-05-12 US disclosed
US-20080234346-A1 PYRAZALIDINONE COMPOUNDS AS LIGANDS OF THE PROSTAGLANDIN EP2 AND/OR EP4 RECEPTORS LABORATOIRES SERONO S.A. (CH) 2008-09-25 US disclosed
US-7410991-B2 Pyrazolidinone compounds as ligands of the prostaglandin EP2 and/or EP4 receptors LABORATOIRES SERONO S.A. (CH) 2008-08-12 US disclosed
EP-1847533-A1 SIX-MEMBERED HETEROCYCLIC COMPOUND AND THE USE THEREOF Asahi Kasei Pharma Corporation (JP) 2007-10-24 EP disclosed
US-20070060590-A1 6-Membered heterocyclic compound and use thereof ASAHI KASEI PHARMA CORPORATION (JP) 2007-03-15 US disclosed
EP-1244661-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PAIN AstraZeneca AB (SE) 2002-10-02 EP disclosed
WO-2001047926-A1 COMPOUNDS AND METHODS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2001-07-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080234346-A1 PYRAZALIDINONE COMPOUNDS AS LIGANDS OF THE PROSTAGLANDIN EP2 AND/OR EP4 RECEPTORS PTGER4, PTGER2, PTGER1 CYP4A11 130/4885CYP4F2 385/4885LOXL2 1792/4885
US-20070060590-A1 6-Membered heterocyclic compound and use thereof WNT1, CYP11B2, CYP11B1 CYP4A11 56/4885CYP4F2 781/4885LOXL2 183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.