SCHEMBL4079372

SCHEMBL4079372

O=C1C=C(Cc2cccc(Cl)c2)C(=O)N1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DAO P14920 3/20 0.48
PNMT P11086 1/20 0.42
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HCAR2 Q8TDS4 1/20 0.40
PNP P00491 1/20 0.40
TAAR1 Q96RJ0 2/20 0.40
MAOA P21397 1/20 0.40
MAOB P27338 1/20 0.40
CYP3A4 P08684 1/20 0.39
IDO1 P14902 1/20 0.39
AGXT P21549 1/20 0.39
C3AR1 Q16581 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL549018 0.88 MAOA (0.35) DAOMAOAMAOB
SCHEMBL3729851 0.81 DAO (0.48) DAOTAAR1CYP3A4IDO1
SCHEMBL94148 0.79 MAOA (0.48) DAOMAOAMAOB
Ammonia Solution, Strong SCHEMBL27962960 0.78 MAOA (0.47) DAOMAOAMAOB
SCHEMBL3669619 0.77 CMA1 (0.48) DAOTAAR1IDO1AGXT
SCHEMBL9508340 0.77 MAOA (0.35) MAOAMAOB
Ethylene SCHEMBL28271283 0.76 MAOA (0.46) DAOMAOAMAOB
SCHEMBL18972983 0.75 AGXT (0.46) TAAR1CYP3A4AGXT
SCHEMBL18972987 0.75 TDP2 (0.38)
SCHEMBL28232297 0.74 DAO (0.39) DAOMAPTPNPMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1874298-A4 METHODS AND COMPOSITIONS FOR PRODUCTION, FORMULATION AND USE OF 1-ARYL-3-AZABICYCLO[3,1,0]HEXANES DOV PHARMACEUTICAL INC (US) 2009-08-05 EP disclosed
EP-1874298-A2 METHODS AND COMPOSITIONS FOR PRODUCTION, FORMULATION AND USE OF 1-ARYL-3-AZABICYCLO[3,1,0]HEXANES DOV Pharmaceutical Inc. (US) 2008-01-09 EP disclosed
WO-2006096810-A2 METHODS AND COMPOSITIONS FOR PRODUCTION, FORMULATION AND USE OF 1-ARYL-3-AZABICYCLO[3.1.0] HEXANES DOV PHARMACEUTICAL, INC. (US) 2006-09-14 WO disclosed