SCHEMBL4080097

SCHEMBL4080097

Oc1c(C(O)C2CCN(c3ncccn3)CC2)ccc(-c2ccccc2)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A7 Q99884 3/20 0.40
KDM4E B2RXH2 6/20 0.39
ALDH1A1 P00352 3/20 0.39
TSHR P16473 3/20 0.39
CYP2C19 P33261 1/20 0.39
HTR1A P08908 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 2/20 0.36
MAPT P10636 1/20 0.36
GAA P10253 1/20 0.36
HTT P42858 1/20 0.36
CSNK1D P48730 1/20 0.35
MAPK14 Q16539 1/20 0.35
RIPK1 Q13546 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3828015 0.85 KDM4E (0.38) SLC6A7KDM4EALDH1A1TSHRCYP2C19
SCHEMBL3893682 0.82 KDM4E (0.40) SLC6A7KDM4EALDH1A1TSHRCYP2C19
SCHEMBL3812208 0.80 ALDH1A1 (0.44) SLC6A7KDM4EALDH1A1TSHRCYP2C19
SCHEMBL3832885 0.79 HTR1A (0.41) SLC6A7KDM4EALDH1A1TSHRCYP2C19
SCHEMBL4234602 0.75 SLC6A7 (0.50) SLC6A7
SCHEMBL4497275 0.75 SLC6A7 (0.50) SLC6A7
SCHEMBL4234609 0.75 SLC6A7 (0.50) SLC6A7
SCHEMBL4078446 0.74 ALDH1A1 (0.41) SLC6A7KDM4EALDH1A1TSHRCYP2C19
SCHEMBL3832888 0.74 MEN1 (0.45) SLC6A7KDM4EALDH1A1TSHRCYP2C19
SCHEMBL4075764 0.72 ESR2 (0.36) SLC6A7ALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2084145-A2 (S)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM AND METHODS OF THEIR USE Lexicon Pharmaceuticals, Inc. (US) 2009-08-05 EP claimed
WO-2008067120-A2 (S)-PHENYL(HETEROCYCLE)METHANOL-BASED COMPOUNDS, COMPOSITIONS COMPRISING THEM AND METHODS OF THEIR USE LEXICON PHARMACEUTICALS, INC. (US) 2008-06-05 WO claimed